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Antibody

6.5 - 270 kDa 범위를 커버하는 3가지 컬러 밴드를 포함하며,
최대 100%까지의 transfer 효과를 개런티하는 Prestained protein ladder를 소개합니다.

CNS Target LeadHunter Panel (#PP280)  

  • CNS 연구에 관련된 94가지 assay를 제공합니다. 
  • Receptors, ionic channels, transporters, nuclear hormone receptors, enzyme에 대한 스크리닝 결과를 제공합니다.
  • Test Sample Requirements: 210 μl of a 10 mM stock or 1.5 mg pre-weighed powder (assuming FW≦500 and purity 100%)

 

GPCR   Ion Channel
200510 Adenosine A1   214510 Calcium Channel L-Type, Benzothiazepine
200610 Adenosine A2A   214600 Calcium Channel L-Type, Dihydropyridine
200650 Adenosine A2B   215000 Calcium Channel L-Type, Phenylalkylamine
200720 Adenosine A3   216000 Calcium Channel N-Type
203110 Adrenergic alpha1A   226810 GABAA, Chloride Channel, TBOB
203210 Adrenergic alpha1B   226600 GABAA, Flunitrazepam, Central
203630 Adrenergic alpha2A   232600 Glutamate, AMPA
203710 Adrenergic alpha2B   232710 Glutamate, Kainate
203810 Adrenergic alpha2C   232810 Glutamate, NMDA, Agonism
204010 Adrenergic beta1   233000 Glutamate, NMDA, Phencyclidine
204110 Adrenergic beta2   239000 Glycine, Strychnine-Sensitive
212620 Bradykinin B2   299031 Nicotinic Acetylcholine alpha4beta2, Cytisine
214020 Calcitonin Gene-Related Peptide CGRP1   299032 Nicotinic Acetylcholine alpha7, Bungarotoxin
217050 Cannabinoid CB1   265800 Potassium Channel [SKCA]
217100 Cannabinoid CB2   299036 Purinergic P2X
218030 Cholecystokinin CCK1 (CCKA)   271910 Serotonin (5-Hydroxytryptamine) 5-HT3
218130 Cholecystokinin CCK2 (CCKB)   279510 Sodium Channel, Site 2
219500 Dopamine D1   Nuclear Hormone Receptor
219600 Dopamine D2L   206000 Androgen (Testosterone)
219800 Dopamine D3   226010 Estrogen ERalpha
220000 Dopamine D4.4   232030 Glucocorticoid
224010 Endothelin ETA   Transporter
228710 GABAB1B   202000 Transporter, Adenosine
237000 Glutamate, Metabotropic, mGlu5   204410 Transporter, Norepinephrine (NET)
239610 Histamine H1   220320 Transporter, Dopamine (DAT)
239820 Histamine H3   226400 Transporter, GABA
251600 Melatonin MT1   274030 Transporter, Serotonin (5-Hydroxytryptamine) (SERT)
252610 Muscarinic M1   Enzyme
252710 Muscarinic M2   107710 ATPase, Na+/K+, Heart, Pig
252810 Muscarinic M3   112020 Carbonic Anhydrase II
252910 Muscarinic M4   199019 Catechol-O-Methyl Transferase (COMT)
253010 Muscarinic M5   104010 Cholinesterase, Acetyl, ACES
255520 Tachykinin NK1   118050 CYP450, 1A2
257010 Neuropeptide Y Y1   118070 CYP450, 2C19
257110 Neuropeptide Y Y2   118080 CYP450, 2D6
260130 Opiate delta1 (OP1, DOP)   118090 CYP450, 3A4
260210 Opiate kappa (OP2, KOP)   199015 GABA Transaminase
260430 Opiate mu (OP3, MOP) [3H]morphine   140010 Monoamine Oxidase MAO-A
299002 Orexin OX2   140120 Monoamine Oxidase MAO-B
299030 Orexin OX1   107310 Peptidase, Angiotensin Converting Enzyme
260900 Oxytocin   112250 Peptidase, CTSB (Cathepsin B)
271110 Serotonin (5-Hydroxytryptamine) 5-HT1A   112650 Peptidase, CTSL (Cathepsin L)
271230 Serotonin (5-Hydroxytryptamine) 5-HT1B   154420 Phosphodiesterase PDE4D2
271650 Serotonin (5-Hydroxytryptamine) 5-HT2A   176610 Protein Serine/Threonine Kinase, MAPK14 (p38alpha)
271700 Serotonin (5-Hydroxytryptamine) 5-HT2B   170020 Protein Tyrosine Kinase, EGF Receptor
271800 Serotonin (5-Hydroxytryptamine) 5-HT2C   174990 Protein Tyrosine Kinase, Insulin Receptor
272320 Serotonin (5-Hydroxytryptamine) 5-HT7   195010 Tyrosine Hydroxylase
287530 Vasopressin V1A   Mitochondrial Function
      299008 BZDp (TSPO)
      Transmembrane
      278300 Sigma, Non-Selective

 

 

  

Drug Abuse Safety SafetyScreen Panel (#PP279) 

  • Drug Abuse (약물남용)에 관련된 48가지 assay 실험을 제공합니다.  
  • FDA의 Assessment of Abuse Potential of Drugs 가이드라인에 따른 시험법을 준수합니다. 
  • Dopamine, Serotonin, GABA, Opioid, Cannabinoid, NMDA, Ion channel complex (calcium, potassium, chloride등), transporter 타겟에 대해 검증합니다.  
  • Test Sample Requirements:120 μl of a 10 mM stock or 1 mg pre-weighed powder (assuming FW≦500 and purity 100%)

 

GPCR   Enzyme
203110 Adrenergic alpha1A   104010 Cholinesterase, Acetyl, ACES
203210 Adrenergic alpha1B   195010 Tyrosine Hydroxylase
203400 Adrenergic alpha1D   Ion Channel
203630 Adrenergic alpha2A   216000 Calcium Channel N-Type
203710 Adrenergic alpha2B   226600 GABAA, Flunitrazepam, Central
203810 Adrenergic alpha2C   232600 Glutamate, AMPA
204010 Adrenergic beta1   232710 Glutamate, Kainate
204110 Adrenergic beta2   232810 Glutamate, NMDA, Agonism
217050 Cannabinoid CB1   233000 Glutamate, NMDA, Phencyclidine
217100 Cannabinoid CB2   299032 Nicotinic Acetylcholine alpha7, Bungarotoxin
219500 Dopamine D1   258660 Nicotinic Acetylcholine alpha7, Methyllycaconitine
219700 Dopamine D2S   271910 Serotonin (5-Hydroxytryptamine) 5-HT3
228610 GABAB1A   Nuclear Hormone Receptor
228710 GABAB1B   226010 Estrogen ERalpha
236400 Glutamate, Metabotropic, mGlu2   226050 Estrogen ERbeta
252610 Muscarinic M1   232030 Glucocorticoid
252710 Muscarinic M2   Transporter
252810 Muscarinic M3   220320 Transporter, Dopamine (DAT)
252910 Muscarinic M4   226400 Transporter, GABA
253010 Muscarinic M5   204410 Transporter, Norepinephrine (NET)
260130 Opiate delta1 (OP1, DOP)   274030 Transporter, Serotonin (5-Hydroxytryptamine) (SERT)
260210 Opiate kappa (OP2, KOP)      
260430 Opiate mu (OP3, MOP) [3H]morphine      
299030 Orexin OX1      
299002 Orexin OX2      
271110 Serotonin (5-Hydroxytryptamine) 5-HT1A      
271230 Serotonin (5-Hydroxytryptamine) 5-HT1B      
271650 Serotonin (5-Hydroxytryptamine) 5-HT2A      
271700 Serotonin (5-Hydroxytryptamine) 5-HT2B      
271800 Serotonin (5-Hydroxytryptamine) 5-HT2C      

 

  

  

Pain Target LeadHunter Panel (#PP273) 

  • Pain target에 관련된 44가지 assay 실험을 제공합니다.  
  • 모든 유형의 통증과 관련있는 GPCR, Ion channel, neurotransmitter, transporter, enzyme에 대한 스크리닝을 제공합니다. 
  • 통증치료에 대한 진통제 발굴 및 연구에 유용합니다. 
  • Test Sample Requirements: 120 μl of a 10 mM stock or 1 mg pre-weighed powder (assuming FW≦500 and purity 100%)

 

GPCR   Enzyme
200720 Adenosine A3   116030 Cyclooxygenase COX-1
203110 Adrenergic alpha1A   118030 Cyclooxygenase COX-2
203630 Adrenergic alpha2A   199008 Fatty Acid Amide Hydrolase (FAAH)
203810 Adrenergic alpha2C   142000 Nitric Oxide Synthase, Neuronal (nNOS)
210120 Angiotensin AT2   176610 Protein Serine/Threonine Kinase, MAPK14 (p38alpha)
212520 Bradykinin B1   175040 Protein Tyrosine Kinase, NTRK1 (TRKA)
212620 Bradykinin B2   Ion Channel
214020 Calcitonin Gene-Related Peptide CGRP1   216020 Calcium Channel Cav2.2, [3H]Gabapentin
217050 Cannabinoid CB1   226600 GABAA, Flunitrazepam, Central
217100 Cannabinoid CB2   232810 Glutamate, NMDA, Agonism
217550 Chemokine CCR2B   232910 Glutamate, NMDA, Glycine
239820 Histamine H3   233000 Glutamate, NMDA, Phencyclidine
258010 Neurotensin NT1   258730 Nicotinic Acetylcholine alpha3beta4
260130 Opiate delta1 (OP1, DOP)   258660 Nicotinic Acetylcholine alpha7, Methyllycaconitine
260210 Opiate kappa (OP2, KOP)   299036 Purinergic P2X
260410 Opiate mu (OP3, MOP)   271910 Serotonin (5-Hydroxytryptamine) 5-HT3
268110 Prostanoid EP1   279510 Sodium Channel, Site 2
268200 Prostanoid EP2   Transporter
299006 Prostanoid EP3   204410 Transporter, Norepinephrine (NET)
268420 Prostanoid EP4   274030 Transporter, Serotonin (5-Hydroxytryptamine) (SERT)
268820 Purinergic P2Y, Non-Selective   Transmembrane
271110 Serotonin (5-Hydroxytryptamine) 5-HT1A   299034 Sigma1
271230 Serotonin (5-Hydroxytryptamine) 5-HT1B  
272320 Serotonin (5-Hydroxytryptamine) 5-HT7  
255520 Tachykinin NK1      

 

   

Neurodegeneration Phenotypic LeadHunter Panel (#PP283)  

  •  가장 흔한 신경퇴행성 질환인 알츠하이머병(AD)과 파킨슨병(PD)의 잠재적 화합물을 스크리닝하기 위한 3가지 cell-based assay 실험을 제공합니다.
  • 가족성 AD의 β-amyloid/과인산화 tau, 산발성 AD의 APOE4, PD 진행과 관련된 α-synuclein을 포함한 유전적 변이 관련 신경변성을 확인합니다. 
  • Test Sample Requirements: 240 μl of a 10 mM stock or 1.5 mg pre-weighed powder (assuming FW≦500 and purity 100%) 

 

Family
Name
Item
Protein
Organism
Assay Sub Type
Cell Based Phenotypic Alpha-Synuclein A53T Parkinson’s Disease Genetic Cell Based Agonist Neurite Outgrowth Assay, Panlabs 332400-0 SYUA_HUMAN Human Cell Based
Cell Based Phenotypic APOEε4 C130R Sporadic Alzheimer’s Disease Genetic Cell Based Agonist Neurite Outgrowth Assay, Panlabs 332440-0 APOE_HUMAN Human Cell Based
Cell Based Phenotypic APP- PS1- MAPT Familial Alzheimer’s Disease Genetic Cell Based Agonist Neurite Outgrowth Assay, Panlabs 332460-0 A4_HUMAN Human Cell Based

 

  

Alzheimer's MoA LeadHunter Panel (#PP284)

  • 신경전달, 글루타메이트 흥분독성, β-아밀로이드의 bioprocess, 타우 과인산화 및 신경염증을 포함한 MoA 기반 표적을 사용합니다.
  • 알츠하이머 치료제 discovery를 위한 41가지 assay를 제공합니다. 
  • Test Sample Requirements: 120 μl of a 10 mM stock or 1 mg pre-weighed powder (assuming FW≦500 and purity 100%)

 

Neurotransmission   Disease-modifying
Cholinergic   Glutamate Excitotoxicity
104010 AChE   279450 279510 Nav
104050 BuChE   200610 Adenosine A2AR
252610 M1   232600 AMPAR
258660 α7nAChR   237000 mGlu5
Monoaminergic   234000 NMDAR-ifenprodil
140010 MAO-A   233010 NMDAR-MK801
140120 MAO-B   299034 σ1R
199019 COMT   299007 σ2R
Serotonergic   b-amyloid
271120 5-HT1A   164700 BACE-1
272000 5-HT4   163950 ECE-1
272200 5-HT6   164010 NEP
Histaminergic   282910 SST4
239820 H3R   Phospho-tau
GABA   168040 CAMK2D
226630 GABA-A   172020 FYN
226400 GABA transporter   176500 GSK-3β
      176610 p38-MAPK
      Neuroinflammation
      199020 15-LO
      112250 CathB
      116030 COX-1
      118030 COX-2
      244600 CX3CR1
      189240 dusp22
      199008 FAAH
      125810 IDO
      199010 iNOS 
      121000 mpo
      299037 PAF

   

 

Parkinson's MoA LeadHunter Panel (#PP285)   

  • 파킨슨병(PD)은 운동 장애를 특징으로 하는 진행성 신경퇴행성 질환입니다. Lewy body inclusion 및 진행성 도파민성 신경 세포 손실은 PD의 병리학적 특징입니다.
  • PP285에는 메커니즘의 다중 프로필을 이해하기 위해 도파민성 및 비도파민성 수용체, 수송체, 이온 채널, 운동 및 비운동 결손과 관련된 효소 분석 등, 27가지 assay를 제공합니다.
  • Test Sample Requirements:120 μl of a 10 mM stock or 1 mg pre-weighed powder (assuming FW≦500 and purity 100%)  

 

Motor   Non-Motor
200610 Adenosine A2AR   271120 5-HT1A
232600 AMPAR   271230 5-HT1B
216010 Cav2.2   271650 5-HT2A
199019 COMT   104010 AChE
219500 D1   104050 BuChE
219600 D2L   239820 H3R
219700 D2S   279450 Nav
219800 D3   274030 SET
220000 D4.4   299034 σ1R
220100 D4.7   299007 σ2R
220200 D5      
220320 DAT      
141010 MAO-A      
140120 MAO-B      
237000 mGlu5      
234000 NMDAR-ifenprodil      
233010 NMDAR-MK801      

 

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0.5 ml Elite Pre-stained Protein Ladder (2 x 0.25 ml) PAL-EPL-500 0.5ml 500
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