도파민 수용체 연구 | GPCR Dopamine Receptor Agonist & Antagonist

시약 및 기기 상세

도파민 수용체 연구 | GPCR Dopamine Receptor Agonist & Antagonist

D1, D2, D3, D4, D5 Dopamine receptor 연구에 필요한 small molecule을 소개합니다.

프린트 제품 문의

특징

Dopamine은 포유동물의 뇌에 존재하는 주요 catecholamine neurotransmitter로, 운동, 신경내분비, 인지 및 감정을 포함한 다양한 기능을 담당합니다. Dopamine은 또한 catecholamine 방출, 호르몬 분비, 위장 운동을 포함한 다양한 다른 과정을 조절하는 역할을 합니다.
D1, D2, D3, D4, D5 Dopamine receptor에 대한 agonist, antagonist를 제공합니다.

주요 제품

D1 and D5 Receptors Agonists & Antagonists
Cat. No.	Product	Activity
2073	(R)-(-)-Apomorphine hydrochloride	Dopamine agonist; non-subtype-selective
1534	A 68930 hydrochloride	Potent and selective D1-like agonist
1701	A 77636 hydrochloride	Potent and selective D1-like agonist; orally active
1249	CY 208-243	Selective D1-like agonist
0884	Dihydrexidine hydrochloride	Selective D1-like agonist
3548	Dopamine hydrochloride	Endogenous agonist at dopamine D1-5 receptors
1659	Fenoldopam hydrochloride	Selective D1-like partial agonist
1674	LE 300	Potent and selective D1 antagonist
3992	NPEC-caged-dopamine	Caged version of dopamine (Cat. No. 3548)
0925	SCH 23390 hydrochloride	Selective D1-like antagonist; also 5-HT2C agonist and Kir3 channel blocker
2299	SCH 39166 hydrobromide	High affinity D1-like antagonist
0922	SKF 38393 hydrobromide	Selective D1-like agonist
1662	SKF 77434 hydrobromide	Selective D1-like partial agonist
1447	SKF 81297 hydrobromide	D1 agonist
5719	SKF 82958 hydrobromide	D1 agonist
1586	SKF 83566 hydrobromide	Potent and selective D1-like antagonist; also inhibits adenylyl cyclase 2
2075	SKF 83822 hydrobromide	Selective D1-like agonist
2074	SKF 83959 hydrobromide	D1-like partial agonist

D2 Receptors Agonists & Antagonists
Cat. No.	Product	Activity
0775	(+)-UH 232 maleate	D2 autoreceptor antagonist. Also D3 partial agonist
5584	Aripiprazole	High affinity D2 and 5-HT1A receptor partial agonist; also 5-HT2A antagonist
2759	B-HT 920	D2 agonist; also α2-adrenoceptor agonist and 5-HT3 antagonist
5858	Droperidol	D2 antagonist
3940	GSK 789472 hydrochloride	D2 partial agonist; D3 antagonist
1003	L-741,626	High affinity D2 antagonist
2495	Melperone hydrochloride	D2 antagonist; also 5-HT2A antagonist; neuroleptic
6171	MLS 1547	G protein-biased D2 partial agonist
4349	Olanzapine	D2 antagonist; also 5-HT2A antagonist; atypical antipsychotic
4493	Paliperidone	D2 antagonist; also 5-HT2A antagonist; atypical antipsychotic
5041	PAOPA	Allosteric modulator of D2 receptors
3287	Prochlorperazine dimaleate	D2 receptor antagonist; also 5-HT3 and nAChR antagonist
4735	Quetiapine hemifumarate	D2 antagonist; also 5-HT2 antagonist; atypical antipsychotic
2865	Risperidone	D2 antagonist; also 5-HT2A antagonist; atypical antipsychotic
3896	Rotigotine hydrochloride	D2 and D3 agonist
2773	Sumanirole maleate	Selective D2 agonist
3085	Ziprasidone hydrochloride	D2 antagonist; also 5-HT2A antagonist; atypical antipsychotic
3996	Zotepine	D2 antagonist; also 5-HT2A and H1 antagonist; atypical antipsychotic

D3 Receptors Agonists & Antagonists
Cat. No.	Product	Activity
1243	(+)-PD 128907 hydrochloride	High affinity D3 agonist (D3 ≥ D2 > D4)
0706	7-Hydroxy-DPAT hydrobromide	Dopamine agonist (D3 ≥ D2 < > D4)
1847	Eticlopride hydrochloride	D3 antagonist (D3 > D2)
3940	GSK 789472 hydrochloride	D3 antagonist. Also D2 partial agonist
1347	Nafadotride	Highly potent, preferential D3 antagonist
2635	NGB 2904	Potent and selective D3 antagonist
3887	PG 01037 dihydrochloride	Selective D3 antagonist
3355	PNU 177864 hydrochloride	Highly selective D3 antagonist
4174	Pramipexole dihydrochloride	Selective D3 agonist
3896	Rotigotine hydrochloride	D2 and D3 agonist
4207	SB 277011A dihydrochloride	Selective D3 antagonist
1357	U 99194 maleate	Potent and selective D3 antagonist

D4 Receptors Agonists & Antagonists
Cat. No.	Product	Activity
4552	A 412997 dihydrochloride	Selective D4 agonist
2214	ABT 724 trihydrochloride	Potent and selective D4 partial agonist; proerectile
2645	Fananserin	D4 antagonist; also 5-HT2A antagonist
1004	L-741,742 hydrochloride	Highly selective D4 antagonist
1002	L-745,870 trihydrochloride	Highly selective D4 antagonist
3298	NGD 94-1	Selective D4 receptor ligand
1065	PD 168077 maleate	High affinity, selective D4 agonist
3529	PD 168568 dihydrochloride	Potent and selective D4 antagonist
2735	PNU 96415E	D4 and 5-HT2A antagonist; antipsychotic
2329	Ro 10-5824 dihydrochloride	Selective D4 partial agonist
4185	Sonepiprazole	Selective D4 antagonist
4380	WAY 100635 maleate	D4 agonist; also potent 5-HT1A antagonist

Dopamine Transporters Inhibitors
Cat. No.	Product	Activity
2148	(±)-McN 5652	Potent, orally active 5-HT uptake inhibitor. Also inhibits noradrenalin and dopamine uptake in vitro
3027	(±)-MDMA hydrochloride	Inhibitor of dopamine and 5-HT uptake; hallucinogenic
6131	(R)-Modafinil	Dopamine uptake inhibitor
4798	(S)-Duloxetine hydrochloride	Potent 5-HT and NA reuptake inhibitor; also blocks dopamine reuptake
0917	3-CPMT	Dopamine uptake inhibitor
0918	3α-Bis-(4-fluorophenyl) methoxytropane hydrochloride	Potent dopamine uptake inhibitor
4946	AIM 100	Promotes endocytosis and oligomerization of DAT; also Ack1 inhibitor
4357	Bicifadine hydrochloride	Noradrenalin, 5-HT and dopamine re-uptake inhibitor
2831	Bupropion hydrochloride	Non-selective inhibitor of dopamine and noradrenalin transporters
2833	Cocaine hydrochloride	Inhibitor of monoamine transporters
5200	FFN 102 mesylate	Selective fluorescent substrate of DAT and VMAT2
0513	GBR 12783 dihydrochloride	Potent and selective DA uptake inhibitor
0421	GBR 12909 dihydrochloride	Selective DA uptake inhibitor; also σ ligand
0514	GBR 12935 dihydrochloride	Selective dopamine uptake inhibitor
0420	GBR 13069 dihydrochloride	Potent dopamine uptake inhibitor
1588	Indatraline hydrochloride	Potent dopamine uptake inhibitor; also inhibits 5-HT and noradrenalin uptake
4351	JHW 007 hydrochloride	High affinity dopamine uptake inhibitor
1992	Nomifensine	Potent noradrenalin and dopamine uptake inhibitor. Antidepressant
2742	Reserpine	Inhibitor of vesicular monoamine transport
1497	Rimcazole dihydrochloride	DAT inhibitor. Also σ2 antagonist
2175	Tetrabenazine	Potent inhibitor of vesicular monoamine transport; depletes dopamine stores
1812	Threo-methylphenidate hydrochloride	Inhibitor of dopamine and noradrenalin transporters. Psychomotor stimulant

Non-Selective Dopamine Agonists & Antagonists
Cat. No.	Product	Activity
1061	(-)-Quinpirole hydrochloride	Selective D2-like agonist
0678	(+)-AJ 76 hydrochloride	Antagonist; preferential action at D2-like autoreceptors
0775	(+)-UH 232 maleate	D2 autoreceptor antagonist. Also D3 partial agonist
2073	(R)-(-)-Apomorphine hydrochloride	Dopamine agonist; non-subtype-selective
0894	(RS)-(±)-Sulpiride	Standard selective D2-like antagonist
0895	(S)-(-)-Sulpiride	Standard selective D2-like antagonist
0782	2-CMDO	D2-like antagonist; displays some D4 selectivity
0701	3'-Fluorobenzylspiperone maleate	D2-like receptor ligand
0524	AMI-193	D2-like antagonist; also selective 5-HT2 antagonist
2132	Amisulpride	Selective D2 and D3 antagonist; atypical antipsychotic
3737	Asenapine maleate	Non-selective 5-HT, dopamine, adrenalin and histamine receptor antagonist; antipsychotic agent
0427	Bromocriptine mesylate	D2-like agonist (D2>D3>D4)
2664	Cabergoline	D2-like agonist (D2>D3>D4)
2193	Carmoxirole hydrochloride	Selective, peripherally acting D2-like agonist
0444	Clozapine	Dopamine antagonist with some D4 selectivity; also 5-HT2A/2C antagonist
0474	Dihydroergocristine mesylate	Dopamine partial agonist; also adrenergic partial agonist and 5-HT antagonist
0475	Dihydroergotamine mesylate	D2-like partial agonist; also α-adrenergic partial agonist and 5-HT antagonist
2536	Domperidone	Peripheral D2-like antagonist
3548	Dopamine hydrochloride	Endogenous agonist at dopamine D1-5 receptors
1847	Eticlopride hydrochloride	D2 and D3 antagonist (D3 > D2)
4057	Flupenthixol dihydrochloride	Dopamine antagonist
0931	Haloperidol hydrochloride	Dopamine antagonist; displays some D2 selectivity
3788	L-DOPA	Dopamine precursor
4052	Lisuride maleate	Dopamine agonist; antiparkinson's agent
1644	Mesulergine hydrochloride	D2-like partial agonist; also 5-HT2A and 5-HT2C antagonist
1746	Nemonapride	Highly potent D2-like antagonist; also 5-HT1A agonist
3992	NPEC-caged-dopamine	Caged dopamine
0937	Pimozide	D2-like antagonist; also high affinity 5-HT7 antagonist
1031	Piribedil dihydrochloride	Dopamine agonist
1519	Quinelorane hydrochloride	D2 and D3 agonist
1810	Raclopride	Potent and selective D2 and D3 antagonist
0916	Remoxipride hydrochloride	Selective D2-like antagonist
3680	Ropinirole	Selective D2-like agonist
1559	Roxindole hydrochloride	Dopamine D2 autoreceptor agonist. Also has affinity for D3, D4, 5-HT1A receptors and the 5-HT transporter
0995	Spiperone hydrochloride	D2-like antagonist; also 5-HT2A antagonist
3070	Thioridazine hydrochloride	Dopamine receptor antagonist; antipsychotic

Vesicular Monoamine Transporters Inhibitors
Cat. No.	Product	Activity
5200	FFN 102 mesylate	Selective fluorescent substrate of VMAT2 and DAT
5911	FFN 200 dihydrochloride	Selective fluorescent VMAT2 substrate
5043	FFN 206 dihydrochloride	Fluorescent VMAT2 substrate
6717	FFN 270	Fluorescent substrate for NET and VMAT2
3878	FFN 511	Fluorescent substrate for VMAT2
2742	Reserpine	Inhibitor of vesicular monoamine transport
5168	Rose Bengal	Potent VGlut and VMAT inhibitor; cell permeable
2175	Tetrabenazine	Potent inhibitor of vesicular monoamine transport

주문정보

주문정보 - Cat No, PRODUCT, SIZE, 수량 등 항목으로 구성되어있습니다.
Product	Cat.No.	Size	Maker
(RS)-(+/-)-Sulpiride (100 mg)	0894	100 mg	TOCRIS
(S)-(-)-Sulpiride (100 mg)	0895	100 mg	TOCRIS
A 77636 hydrochloride (10 mg)	1701	10 mg	TOCRIS
A 77636 hydrochloride (50 mg)	1701	50 mg	TOCRIS
AIM 100 (50 mg)	4946	50 mg	TOCRIS
Asenapine maleate (10 mg)	3737	10 mg	TOCRIS
Asenapine maleate (50 mg)	3737	50 mg	TOCRIS
Bromocriptine mesylate (50 mg)	0427	50 mg	TOCRIS
Cabergoline (10 mg)	2664	10 mg	TOCRIS
Cabergoline (50 mg)	2664	50 mg	TOCRIS
Dihydroergocristine mesylate (100 mg)	0474	100 mg	TOCRIS
Domperidone (50 mg)	2536	50 mg	TOCRIS
Flupenthixol dihydrochloride (50 mg)	4057	50 mg	TOCRIS
Haloperidol hydrochloride (100 mg)	0931	100 mg	TOCRIS
L-DOPA (50 mg)	3788	50 mg	TOCRIS
Lisuride maleate (10 mg)	4052	10 mg	TOCRIS
Lisuride maleate (50 mg)	4052	50 mg	TOCRIS
MLS 1547 (25 MG)	6171	25 mg	TOCRIS
MLS 1547 (5 MG)	6171	5 mg	TOCRIS
NGB 2904 (10 mg)	2635	10 mg	TOCRIS
NGB 2904 (50 mg)	2635	50 mg	TOCRIS
PD 168568 dihydrochloride (10 mg)	3529	10 mg	TOCRIS
PD 168568 dihydrochloride (50 mg)	3529	50 mg	TOCRIS
Pimozide (100 mg)	0937	100 mg	TOCRIS
Quinelorane hydrochloride (10 mg)	1519	10 mg	TOCRIS
Raclopride (10 mg)	1810	10 mg	TOCRIS
Raclopride (50 mg)	1810	50 mg	TOCRIS
Ro 10-5824 dihydrochloride (10 mg)	2329	10 mg	TOCRIS
Ro 10-5824 dihydrochloride (50 mg)	2329	50 mg	TOCRIS
Ropinirole (10 mg)	3680	10 mg	TOCRIS
Ropinirole (50 mg)	3680	50 mg	TOCRIS

전체보기

1
Maker	TOCRIS
Cat.No.	0894
Product	(RS)-(+/-)-Sulpiride (100 mg)
Size	100 mg
Qty
Data Sheet
MSDS

2
Maker	TOCRIS
Cat.No.	0895
Product	(S)-(-)-Sulpiride (100 mg)
Size	100 mg
Qty
Data Sheet
MSDS

3
Maker	TOCRIS
Cat.No.	1701
Product	A 77636 hydrochloride (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

4
Maker	TOCRIS
Cat.No.	1701
Product	A 77636 hydrochloride (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

5
Maker	TOCRIS
Cat.No.	4946
Product	AIM 100 (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

6
Maker	TOCRIS
Cat.No.	3737
Product	Asenapine maleate (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

7
Maker	TOCRIS
Cat.No.	3737
Product	Asenapine maleate (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

8
Maker	TOCRIS
Cat.No.	0427
Product	Bromocriptine mesylate (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

9
Maker	TOCRIS
Cat.No.	2664
Product	Cabergoline (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

10
Maker	TOCRIS
Cat.No.	2664
Product	Cabergoline (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

11
Maker	TOCRIS
Cat.No.	0474
Product	Dihydroergocristine mesylate (100 mg)
Size	100 mg
Qty
Data Sheet
MSDS

12
Maker	TOCRIS
Cat.No.	2536
Product	Domperidone (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

13
Maker	TOCRIS
Cat.No.	4057
Product	Flupenthixol dihydrochloride (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

14
Maker	TOCRIS
Cat.No.	0931
Product	Haloperidol hydrochloride (100 mg)
Size	100 mg
Qty
Data Sheet
MSDS

15
Maker	TOCRIS
Cat.No.	3788
Product	L-DOPA (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

16
Maker	TOCRIS
Cat.No.	4052
Product	Lisuride maleate (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

17
Maker	TOCRIS
Cat.No.	4052
Product	Lisuride maleate (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

18
Maker	TOCRIS
Cat.No.	6171
Product	MLS 1547 (25 MG)
Size	25 mg
Qty
Data Sheet
MSDS

19
Maker	TOCRIS
Cat.No.	6171
Product	MLS 1547 (5 MG)
Size	5 mg
Qty
Data Sheet
MSDS

20
Maker	TOCRIS
Cat.No.	2635
Product	NGB 2904 (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

21
Maker	TOCRIS
Cat.No.	2635
Product	NGB 2904 (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

22
Maker	TOCRIS
Cat.No.	3529
Product	PD 168568 dihydrochloride (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

23
Maker	TOCRIS
Cat.No.	3529
Product	PD 168568 dihydrochloride (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

24
Maker	TOCRIS
Cat.No.	0937
Product	Pimozide (100 mg)
Size	100 mg
Qty
Data Sheet
MSDS

25
Maker	TOCRIS
Cat.No.	1519
Product	Quinelorane hydrochloride (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

26
Maker	TOCRIS
Cat.No.	1810
Product	Raclopride (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

27
Maker	TOCRIS
Cat.No.	1810
Product	Raclopride (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

28
Maker	TOCRIS
Cat.No.	2329
Product	Ro 10-5824 dihydrochloride (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

29
Maker	TOCRIS
Cat.No.	2329
Product	Ro 10-5824 dihydrochloride (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

30
Maker	TOCRIS
Cat.No.	3680
Product	Ropinirole (10 mg)
Size	10 mg
Qty
Data Sheet
MSDS

31
Maker	TOCRIS
Cat.No.	3680
Product	Ropinirole (50 mg)
Size	50 mg
Qty
Data Sheet
MSDS

전체보기

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도파민 수용체 연구 | GPCR Dopamine Receptor Agonist & Antagonist | 고마바이오텍

도파민 수용체 연구 | GPCR Dopamine Receptor Agonist & Antagonist

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