| Cyclooxygenase Inhibitors |
| Cat. No. |
Product |
Activity |
| 2796 |
(S)-(+)-Ibuprofen |
Cyclooxygenase
inhibitor (COX-1 > COX-2) |
| 1706 |
Acetaminophen |
Cyclooxygenase inhibitor; may be selective for COX-3 |
| 4092 |
Aspirin |
Cyclooxygenase inhibitor; NSAID |
| 3786 |
Celecoxib |
Selective cyclooxygenase-2 (COX-2) inhibitor |
| 4454 |
Diclofenac
sodium salt |
Cyclooxygenase inhibitor; NSAID |
| 1430 |
DuP 697 |
Cyclooxygenase-2 (COX-2) inhibitor |
| 4522 |
Flufenamic
acid |
Cyclooxygenase inhibitor; NSAID. Also activates TRPC6 |
| 1507 |
FR
122047 hydrochloride |
Cyclooxygenase (COX-1) inhibitor |
| 1708 |
Indomethacin |
Cyclooxygenase inhibitor (COX-1 > COX-2) |
| 2655 |
Naproxen
sodium |
Cyclooxygenase inhibitor |
| 4112 |
Niflumic
acid |
Cyclooxygenase-2 (COX-2) inhibitor; GPR35 agonist |
| 0942 |
NS 398 |
Cyclooxygenase-2 (COX-2) inhibitor |
| 1418 |
Resveratrol |
Cyclooxygenase inhibitor |
| 3919 |
SC 236 |
Selective cyclooxygenase-2 (COX-2) inhibitor |
| 1550 |
SC 560 |
Cyclooxygenase-1 (COX-1) inhibitor |
| 2580 |
Tenidap |
NSAID, cyclooxygenase (COX-1) inhibitor. Also opener of KIR2.3 |
| 4206 |
Valdecoxib |
Selective and potent COX-2 inhibitor |
|
|
|
| Monoamine
Oxidases |
| Cat. No. |
Product |
Activity |
| 1095 |
(R)-(-)-Deprenyl hydrochloride |
MAO-B
inhibitor |
| 3306 |
8-(3-Chlorostyryl)caffeine |
MAO-B inhibitor; also A2A inhibitor |
| 0767 |
Bifemelane
hydrochloride |
Non-selective MAO inhibitor |
| 2460 |
Lazabemide
hydrochloride |
Selective MAO-B inhibitor |
| 6067 |
M
30 dihydrochloride |
Potent and non-selective MAO inhibitor; also an iron chelator
and antioxidant |
| 4395 |
Moclobemide |
Reversible MAO-A inhibitor |
| 0724 |
Pirlindole
mesylate |
MAO-A inhibitor |
| 4308 |
Rasagiline
mesylate |
Selective and irreversible MAO-B inhibitor |
| 3852 |
Tranylcypromine
hydrochloride |
Irreversible and non-selective MAO inhibitor; also inhibits LSD1 |
|
|
|
| Indoleamine 2,3
dioxygenase Inhibitors |
| Cat. No. |
Product |
Activity |
| 5698 |
1-Methyl-D-tryptophan |
Indoleamine
2,3-dioxygenase (IDO) inhibitor |
| 6007 |
INCB
024360-analog |
Potent indoleamine 2,3-dioxygenase (IDO) inhibitor |
|
|
|
| Lipoxygenase
Inhibitors |
| Cat. No. |
Product |
Activity |
| 0645 |
2-TEDC |
5-, 12-,
15-Lipoxygenase inhibitor |
| 1761 |
Baicalein |
5- and 12-Lipoxygenase inhibitor |
| 1311 |
MK 886 |
Inhibitor of 5-lipoxygenase-activating protein (FLAP) |
| 6448 |
ML 351 |
Selective 12/15 LOX inhibitor; active in
vivo |
| 2850 |
PD 146176 |
Selective 15-lipoxygenase inhibitor |
| 3308 |
Zileuton |
5-LOX inhibitor; orally bioavailable |
|
|
|
| Heme Oxygenase |
| Cat. No. |
Product |
Activity |
| 6119 |
OB
24 hydrochloride |
Potent and
selective heme oxygenase 1 (HO-1) inhibitor |
| 0747 |
Tin
protoporphyrin IX dichloride |
Heme oxygenase inhibitor |
|
|
|
| NADPH Oxidases |
| Cat. No. |
Product |
Activity |
| 4663 |
Apocynin |
NADPH-oxidase
inhibitor |
| 0504 |
Diphenyleneiodonium
chloride |
Inhibits NADPH oxidases; also inhibits NOS |
| 6848 |
GSK
2795039 |
NADPH oxidase 2 (NOX2) inhibitor |
| 6654 |
VAS 2870 |
NADPH oxidase (Nox) inhibitor |
|
|
|
| Stearoyl-CoA
9-Desaturase |
| Cat. No. |
Product |
Activity |
| 4845 |
A 939572 |
Potent SCD-1
inhibitor |
| 4847 |
PluriSln 1 |
SCD-1 inhibitor |
|
|
|
| Tryptophan 2,3
dioxygenase Inhibitors |
| Cat. No. |
Product |
Activity |
| 4392 |
680C91 |
Potent and
selective tryptophan 2,3-dioxygenase (TDO) inhibitor |
| 5794 |
LM 10 |
Selective tryptophan 2,3-dioxygenase (TDO) inhibitor |