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Cyclooxygenase
Inhibitors |
|
Cat. No. |
Product
Name |
Activity |
|
2796 |
(S)-(+)-Ibuprofen |
Cyclooxygenase
inhibitor (COX-1 > COX-2) |
|
1706 |
Acetaminophen |
Cyclooxygenase inhibitor; may be selective for COX-3 |
|
4092 |
Aspirin |
Cyclooxygenase inhibitor; NSAID |
|
3786 |
Celecoxib |
Selective cyclooxygenase-2 (COX-2) inhibitor |
|
4454 |
Diclofenac sodium salt |
Cyclooxygenase inhibitor; NSAID |
|
1430 |
DuP 697 |
Cyclooxygenase-2 (COX-2) inhibitor |
|
4522 |
Flufenamic acid |
Cyclooxygenase inhibitor; NSAID. Also activates TRPC6 |
|
1507 |
FR 122047 hydrochloride |
Cyclooxygenase (COX-1) inhibitor |
|
1708 |
Indomethacin |
Cyclooxygenase inhibitor (COX-1 > COX-2) |
|
2655 |
Naproxen sodium |
Cyclooxygenase inhibitor |
|
4112 |
Niflumic acid |
Cyclooxygenase-2 (COX-2) inhibitor; GPR35 agonist |
|
0942 |
NS 398 |
Cyclooxygenase-2 (COX-2) inhibitor |
|
1418 |
Resveratrol |
Cyclooxygenase inhibitor |
|
3919 |
SC 236 |
Selective cyclooxygenase-2 (COX-2) inhibitor |
|
1550 |
SC 560 |
Cyclooxygenase-1 (COX-1) inhibitor |
|
2580 |
Tenidap |
NSAID,
cyclooxygenase (COX-1) inhibitor. Also opener of KIR2.3 |
|
4206 |
Valdecoxib |
Selective and potent COX-2 inhibitor |
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Monoamine Oxidases |
|
Cat. No. |
Product
Name |
Activity |
|
1095 |
(R)-(-)-Deprenyl
hydrochloride |
MAO-B
inhibitor |
|
3306 |
8-(3-Chlorostyryl)caffeine |
MAO-B
inhibitor; also A2A inhibitor |
|
0767 |
Bifemelane hydrochloride |
Non-selective MAO inhibitor |
|
2460 |
Lazabemide hydrochloride |
Selective MAO-B inhibitor |
|
6067 |
M 30 dihydrochloride |
Potent and non-selective MAO inhibitor; also an iron
chelator and antioxidant |
|
4395 |
Moclobemide |
Reversible MAO-A inhibitor |
|
0724 |
Pirlindole mesylate |
MAO-A inhibitor |
|
4308 |
Rasagiline mesylate |
Selective and irreversible MAO-B inhibitor |
|
3852 |
Tranylcypromine hydrochloride |
Irreversible and non-selective MAO inhibitor; also
inhibits LSD1 |
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Indoleamine 2,3 dioxygenase Inhibitors |
|
Cat. No. |
Product
Name |
Activity |
|
5698 |
1-Methyl-D-tryptophan |
Indoleamine
2,3-dioxygenase (IDO) inhibitor |
|
6007 |
INCB 024360-analog |
Potent indoleamine 2,3-dioxygenase (IDO) inhibitor |
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Lipoxygenase Inhibitors |
|
Cat. No. |
Product
Name |
Activity |
|
0645 |
2-TEDC |
5-,
12-, 15-Lipoxygenase inhibitor |
|
1761 |
Baicalein |
5- and 12-Lipoxygenase inhibitor |
|
1311 |
MK 886 |
Inhibitor of 5-lipoxygenase-activating protein (FLAP) |
|
6448 |
ML 351 |
Selective
12/15 LOX inhibitor; active in vivo |
|
2850 |
PD 146176 |
Selective 15-lipoxygenase inhibitor |
|
3308 |
Zileuton |
5-LOX inhibitor; orally bioavailable |
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Monoamine Oxidases |
|
Cat. No. |
Product
Name |
Activity |
|
6119 |
OB 24 hydrochloride |
Potent
and selective heme oxygenase 1 (HO-1) inhibitor |
|
0747 |
Tin protoporphyrin IX dichloride |
Heme oxygenase inhibitor |
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|
|
|
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Monoamine Oxidases |
|
Cat. No. |
Product
Name |
Activity |
|
4663 |
Apocynin |
NADPH-oxidase
inhibitor |
|
0504 |
Diphenyleneiodonium chloride |
Inhibits NADPH oxidases; also inhibits NOS |
|
6848 |
GSK 2795039 |
NADPH oxidase 2 (NOX2) inhibitor |
|
6654 |
VAS 2870 |
NADPH oxidase (Nox) inhibitor |
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Stearoyl-CoA 9-Desaturase |
|
Cat. No. |
Product
Name |
Activity |
|
4845 |
A 939572 |
Potent
SCD-1 inhibitor |
|
4847 |
PluriSln 1 |
SCD-1 inhibitor |
| |
|
|
|
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Tryptophan 2,3 dioxygenase Inhibitors |
|
Cat. No. |
Product
Name |
Activity |
|
4392 |
680C91 |
Potent
and selective tryptophan 2,3-dioxygenase (TDO) inhibitor |
|
5794 |
LM
10 |
Selective tryptophan 2,3-dioxygenase (TDO) inhibitor |