AGC Group (Protein Kinase A,G,C) |
|
Cat. No. |
Product |
Activity |
0741 |
GF 109203X |
Protein kinase C inhibitor |
4143 |
GSK 2334470 |
Highly potent, selective PDPK1 (PDK1) inhibitor |
1288 |
KT 5720 |
Selective protein kinase A inhibitor |
4630 |
SB 747651A dihydrochloride |
Potent MSK1 inhibitor; also inhibits other AGC group kinases |
4635 |
SC 79 |
Akt activator |
|
|
|
CAMK
Group (calcium/calmodulin signaling) |
|
Cat. No. |
Product |
Activity |
5183 |
ETP 45835 dihydrochloride |
Mnk1 and Mnk2 inhibitor |
5134 |
MRT 67307 dihydrochloride |
Salt inducible kinase (SIK) inhibitor; also ULK1 and 2 inhibitor |
5177 |
WZ 4003 |
Potent and selective NUAK1/2 inhibitor |
|
|
|
CK1
Group (Casein Kinase 1) |
|
Cat. No. |
Product |
Activity |
2902 |
D 4476 |
Selective CK1 inhibitor. Also inhibits TGF-βRI |
4281 |
PF 4800567 hydrochloride |
Selective casein kinase 1ε inhibitor |
|
|
|
CMGC
Group (CDK, MAPK, GSK-3, Clks) |
|
Cat. No. |
Product |
Activity |
4753 |
AL 8697 |
Potent and selective p38α inhibitor |
4423 |
CHIR 99021 |
Highly selective GSK-3 inhibitor; acts as Wnt activator |
5095 |
DBM 1285 dihydrochloride |
p38 MAPK inhibitor;
anti-inflammatory |
1202 |
SB 203580 |
Selective inhibitor of p38 MAPK |
1616 |
SB 216763 |
Potent, selective GSK-3 inhibitor |
5040 |
SB 706504 |
p38 MAPK inhibitor |
4875 |
Senexin A |
Cdk8 inhibitor |
3222 |
TCS JNK 6o |
Selective JNK inhibitor |
|
|
|
STE
Group (homologs of yeast sterile 7, sterile 11, sterile 20 kinase) |
Cat. No. |
Product |
Activity |
4842 |
BIX 02189 |
Selective MEK5 and ERK5 inhibitor |
4192 |
PD 0325901 |
Potent inhibitor of MEK1/2 |
1144 |
U0126 |
Potent, selective inhibitor of MEK1 and 2 |
|
|
|
TK
Group (Tyrosine Kinase) |
|
Cat. No. |
Product |
Activity |
5310 |
ASP 3026 |
Potent anaplastic lymphoma kinase (ALK) inhibitor; also potent
ACK inhibitor |
5077 |
DDR1-IN-1 dihydrochloride |
Selective DDR1 inhibitor |
4660 |
KB SRC 4 |
Potent and selective c-Src inhibitor |
5247 |
NVP ADW 742 |
ATP-competitive inhibitor of IGF1R |
3037 |
SU 5416 |
VEGFR inhibitor. Also inhibits KIT, RET, MET and FLT3 |
|
|
|
TKL
Group (Tyrosine kinase-like Kinases) |
|
Cat. No. |
Product |
Activity |
4126 |
DMH-1 |
Selective ALK2 inhibitor |
4986 |
K 02288 |
Type 1 BMP receptor inhibitor |
4745 |
LIMKi 3 |
Potent LIM kinase inhibitor; antitumor |
4945 |
ML 347 |
Potent and selective ALK1 and ALK2 inhibitor |