| Adrenergic α1 Receptors |
|
| Cat. No. |
Product |
Activity |
| 2838 |
(R)-(-)-Phenylephrine hydrochloride |
α1 agonist |
| 1052 |
A 61603 hydrobromide |
α1A agonist |
| 2685 |
Carvedilol |
Potent α1 antagonist; also potent and non-selective β antagonist |
| 0888 |
Cirazoline hydrochloride |
Selective α1 agonist |
| 2964 |
Doxazosin mesylate |
α1 antagonist |
| 0535 |
HEAT hydrochloride |
Highly selective α1 antagonist |
| 0545 |
Ifenprodil hemitartrate |
α1 antagonist. Also NMDA antagonist and σ ligand |
| 0597 |
Naftopidil hydrochloride |
α1 antagonist |
| 0623 |
Prazosin hydrochloride |
α1 and α2B antagonist; also MT3 antagonist |
| 1325 |
RS 100329 hydrochloride |
Potent, subtype-selective α1A antagonist |
| 0985 |
RS 17053 hydrochloride |
α1A antagonist |
| 6663 |
Silodosin |
Selective α1A antagonist |
| 3050 |
Tamsulosin hydrochloride |
Selective α1A antagonist |
| 1506 |
Terazosin hydrochloride |
α1 and α2B antagonist (α1 > α2B). Orally active |
| 6336 |
Trazodone hydrochloride |
5-HT2A and α1 adrenoceptor antagonist; also enhances neural
differentiation |
|
|
|
| Adrenergic
α2 Receptors |
|
| Cat. No. |
Product |
Activity |
| 0928 |
ARC 239 dihydrochloride |
α2B antagonist |
| 2937 |
Atipamezole hydrochloride |
Selective α2 antagonist |
| 2758 |
B-HT 933 dihydrochloride |
Selective α2 agonist |
| 1133 |
BRL 44408 maleate |
Selective α2A antagonist |
| 0690 |
Clonidine hydrochloride |
α2 agonist. Also I1 ligand |
| 2749 |
Dexmedetomidine hydrochloride |
Potent, highly selective α2 agonist. Active isomer of
medetomidine (Cat. No. 5160) |
| 0885 |
Guanabenz acetate |
α2 agonist. Also I2 selective ligand |
| 1030 |
Guanfacine hydrochloride |
α2A agonist |
| 0986 |
Imiloxan hydrochloride |
Highly selective α2B antagonist |
| 2666 |
JP 1302 dihydrochloride |
Potent and selective α2C antagonist |
| 5160 |
Medetomidine hydrochloride |
Potent and highly selective α2 agonist |
| 2018 |
Mirtazapine |
α2 antagonist; also potent 5-HT2, 5-HT3 and H1 antagonist;
antidepressant |
| 0623 |
Prazosin hydrochloride |
α2B and α1 antagonist; also MT3 antagonist |
| 0790 |
Rilmenidine hemifumarate |
I1 ligand. Also α2 agonist. |
| 0987 |
RS 79948 hydrochloride |
Potent and selective α2 antagonist |
| 1324 |
RX 821002 hydrochloride |
Potent, selective α2D antagonist |
| 3866 |
SKF 86466 hydrochloride |
Potent and selective α2 antagonist |
| 3609 |
Tizanidine hydrochloride |
α2 agonist |
| 0425 |
UK 14,304 |
α2 agonist |
| 2466 |
UK 14,304 tartrate |
α2 agonist. Water-soluble form of UK 14,304 (Cat. No. 0425) |
| 1127 |
Yohimbine hydrochloride |
Selective α2 antagonist |
|
|
|
| Adrenergic
β1 Receptors |
|
| Cat. No. |
Product |
Activity |
| 0906 |
Betaxolol hydrochloride |
Selective β1 antagonist |
| 1024 |
CGP 20712 dihydrochloride |
Highly potent and selective β1 antagonist |
| 3256 |
Metoprolol tartrate |
Selective β1 antagonist |
| 3517 |
Nebivolol hydrochloride |
Highly selective β1-adrenoceptor antagonist |
| 0950 |
Xamoterol hemifumarate |
Selective β1 partial agonist |
|
|
|
| Adrenergic
β2 Receptors |
|
| Cat. No. |
Product |
Activity |
| 6219 |
Arformoterol tartrate |
Long-acting β2 agonist (LABA) |
| 1448 |
Formoterol hemifumarate |
Potent and selective β2 agonist |
| 0821 |
ICI 118,551 hydrochloride |
Highly selective β2 inverse agonist |
| 1102 |
Procaterol hydrochloride |
Potent β2 agonist |
| 0634 |
Salbutamol hemisulfate |
β2-adrenoceptor agonist |
| 4712 |
Salmeterol xinafoate |
Long-acting β2 agonist; bronchodilator |
| 1051 |
Zinterol hydrochloride |
Selective β2 agonist |
|
|
|
| Adrenergic
β3 Receptors |
|
| Cat. No. |
Product |
Activity |
| 1060 |
(S)-(-)-Pindolol |
β3 partial agonist; also 5-HT1A and 5-HT1B antagonist; more
active enantiomer of pindolol |
| 0948 |
BRL 37344, sodium salt |
β3 agonist |
| 1134 |
CGP 12177 hydrochloride |
β3 partial agonist. β1/β2 antagonist |
| 1499 |
CL 316243 disodium salt |
Highly selective β3 agonist |
| 2760 |
L-748,337 |
Selective β3 antagonist |
| 2197 |
L-755,507 |
Very potent and selective β3 partial agonist |
| 7070 |
Mirabegron |
Potent and selective β3 agonist |
| 3986 |
SR 58611A hydrochloride |
β3 agonist; displays anxiolytic and antidepressant effects |
| 1511 |
SR 59230A hydrochloride |
Potent and selective β3 antagonist |