Ca2+-ATPase Inhibitors, Activator &
Blockers |
|
Cat. No. |
Product |
Activity |
5869 |
CDN 1163 |
SERCA2 allosteric
activator |
1235 |
Cyclopiazonic acid |
Inhibitor of SERCA
ATPase |
3807 |
Disulfiram |
Reversibly
stimulates SERCA Ca2+-ATPase |
2006 |
Paxilline |
SERCA ATPase
blocker. Also potent BKCa channel blocker |
1138 |
Thapsigargin |
Potent inhibitor of
SERCA ATPase |
|
|
|
Calcium
Binding Protein Antagonists & Inhibitors |
|
Cat. No. |
Product |
Activity |
1688 |
Autocamtide-2-related
inhibitory peptide |
Selective CaM
kinase II inhibitor |
5959 |
Autocamtide-2-related
inhibitory peptide, myristoylated |
CaM kinase II
inhibitor |
2561 |
Calmidazolium
chloride |
Calmodulin
antagonist |
2255 |
CGS 9343B |
Calmodulin
antagonist |
1278 |
KN 93 |
CaM kinase II
inhibitor; also K+ channel blocker (KV) |
1277 |
KN-62 |
CaM kinase II
inhibitor |
0431 |
ML 9 hydrochloride |
Myosin light chain
kinase inhibitor |
1885 |
MLCK inhibitor
peptide 18 |
Selective inhibitor
of myosin light chain kinase |
1551 |
STO-609 acetate |
Selective CaM
kinase kinase inhibitor |
0361 |
W-13 hydrochloride |
Calmodulin
antagonist |
0368 |
W-5 hydrochloride |
Calmodulin
antagonist |
0369 |
W-7 hydrochloride |
Calmodulin
antagonist. Inhibits myosin light chain kinase |
|
|
|
Calcium-Sensing
Receptor Agonists & Antagonists |
|
Cat. No. |
Product |
Activity |
6165 |
AC 265347 |
Biased allosteric
modulator of calcium-sensing receptor (CaSR) |
4387 |
Calhex 231
hydrochloride |
Negative allosteric
modulator of calcium-sensing receptor (CaSR) |
6170 |
Cinacalcet
hydrochloride |
Allosteric
Calcium-sensing receptor (CaSR) agonist |
3626 |
NPS 2143
hydrochloride |
Selective
calcium-sensing receptor (CaSR) antagonist |
3815 |
R 568 hydrochloride |
Positive allosteric
modulator of human calcium-sensing receptor (CaSR) |
|
|
|
Calcium-Sensitive
Protease Inhibitors |
|
Cat. No. |
Product |
Activity |
2950 |
Acetyl-Calpastatin
(184-210) (human) |
Selective
calpain inhibitor |
4863 |
CA 074 |
Selective
cathepsin B inhibitor |
5208 |
E 64 |
Potent
and irreversible cysteine protease inhibitor |
4545 |
E 64d |
Cathepsin
inhibitor; interferes with autolysosomal digestion |
3066 |
L 006235 |
Potent
cathepsin K inhibitor |
1748 |
MG 132 |
Calpain
and proteasome inhibitor |
1269 |
PD 150606 |
Cell
permeable calpain inhibitor |
3625 |
SID 26681509 |
Cathepsin
L inhibitor |
|
|
|
Mitochondrial
Calcium Uniporter Inhibitors |
|
Cat. No. |
Product |
Activity |
3603 |
Kaempferol |
Mitochondrial Ca2+
uniporter (MCU) activator |
1244 |
KB-R7943 mesylate |
Mitochondrial Ca2+
uniporter (MCU) inhibitor |
7195 |
MCU i4 |
Negative modulator
of mitochondrial Ca2+ uniporter (MCU) |