| Ca2+-ATPase Inhibitors, Activator &
Blockers |
|
| Cat. No. |
Product |
Activity |
| 5869 |
CDN 1163 |
SERCA2 allosteric
activator |
| 1235 |
Cyclopiazonic acid |
Inhibitor of SERCA
ATPase |
| 3807 |
Disulfiram |
Reversibly
stimulates SERCA Ca2+-ATPase |
| 2006 |
Paxilline |
SERCA ATPase
blocker. Also potent BKCa channel blocker |
| 1138 |
Thapsigargin |
Potent inhibitor of
SERCA ATPase |
|
|
|
| Calcium
Binding Protein Antagonists & Inhibitors |
|
| Cat. No. |
Product |
Activity |
| 1688 |
Autocamtide-2-related
inhibitory peptide |
Selective CaM
kinase II inhibitor |
| 5959 |
Autocamtide-2-related
inhibitory peptide, myristoylated |
CaM kinase II
inhibitor |
| 2561 |
Calmidazolium
chloride |
Calmodulin
antagonist |
| 2255 |
CGS 9343B |
Calmodulin
antagonist |
| 1278 |
KN 93 |
CaM kinase II
inhibitor; also K+ channel blocker (KV) |
| 1277 |
KN-62 |
CaM kinase II
inhibitor |
| 0431 |
ML 9 hydrochloride |
Myosin light chain
kinase inhibitor |
| 1885 |
MLCK inhibitor
peptide 18 |
Selective inhibitor
of myosin light chain kinase |
| 1551 |
STO-609 acetate |
Selective CaM
kinase kinase inhibitor |
| 0361 |
W-13 hydrochloride |
Calmodulin
antagonist |
| 0368 |
W-5 hydrochloride |
Calmodulin
antagonist |
| 0369 |
W-7 hydrochloride |
Calmodulin
antagonist. Inhibits myosin light chain kinase |
|
|
|
| Calcium-Sensing
Receptor Agonists & Antagonists |
|
| Cat. No. |
Product |
Activity |
| 6165 |
AC 265347 |
Biased allosteric
modulator of calcium-sensing receptor (CaSR) |
| 4387 |
Calhex 231
hydrochloride |
Negative allosteric
modulator of calcium-sensing receptor (CaSR) |
| 6170 |
Cinacalcet
hydrochloride |
Allosteric
Calcium-sensing receptor (CaSR) agonist |
| 3626 |
NPS 2143
hydrochloride |
Selective
calcium-sensing receptor (CaSR) antagonist |
| 3815 |
R 568 hydrochloride |
Positive allosteric
modulator of human calcium-sensing receptor (CaSR) |
|
|
|
| Calcium-Sensitive
Protease Inhibitors |
|
| Cat. No. |
Product |
Activity |
| 2950 |
Acetyl-Calpastatin
(184-210) (human) |
Selective
calpain inhibitor |
| 4863 |
CA 074 |
Selective
cathepsin B inhibitor |
| 5208 |
E 64 |
Potent
and irreversible cysteine protease inhibitor |
| 4545 |
E 64d |
Cathepsin
inhibitor; interferes with autolysosomal digestion |
| 3066 |
L 006235 |
Potent
cathepsin K inhibitor |
| 1748 |
MG 132 |
Calpain
and proteasome inhibitor |
| 1269 |
PD 150606 |
Cell
permeable calpain inhibitor |
| 3625 |
SID 26681509 |
Cathepsin
L inhibitor |
|
|
|
| Mitochondrial
Calcium Uniporter Inhibitors |
|
| Cat. No. |
Product |
Activity |
| 3603 |
Kaempferol |
Mitochondrial Ca2+
uniporter (MCU) activator |
| 1244 |
KB-R7943 mesylate |
Mitochondrial Ca2+
uniporter (MCU) inhibitor |
| 7195 |
MCU i4 |
Negative modulator
of mitochondrial Ca2+ uniporter (MCU) |