Adenosine A1 Receptors Agonist, Antagonist,
Modulators |
Cat. No. |
Product |
Activity |
3576 |
(±)-5'-Chloro-5'-deoxy-ENBA |
Highly selective A1
agonist |
1705 |
2-Chloro-N6-cyclopentyladenosine |
Potent and
selective A1 agonist |
2281 |
2'-MeCCPA |
Highly selective
and potent A1 receptor agonist |
6137 |
8-Cyclopentyl-1,3-dimethylxanthine |
High affinity
adenosine A1 receptor antagonist |
0439 |
DPCPX |
Selective A1
antagonist |
4167 |
KW 3902 |
Selective A1
antagonist |
6863 |
N6-Cyclohexyladenosine |
High affinity A1
receptor agonist |
1702 |
N6-Cyclopentyladenosine |
Potent and
selective A1 agonist |
1363 |
PD 81723 |
Positive allosteric
modulator of A1 receptors |
2465 |
SDZ WAG 994 |
Potent and
selective A1 agonist |
6261 |
VCP 171 |
Positive allosteric
modulator (PAM) of A1 receptors; also allosteric partial agonist in absence
of orthosteric agonist |
|
|
|
Adenosine
A2A Receptor Agonists, Antagonist |
|
Cat. No. |
Product |
Activity |
3306 |
8-(3-Chlorostyryl)caffeine |
Selective A2A
antagonist. Also MAO-B inhibitor |
3937 |
ANR 94 |
Adenosine A2A
antagonist |
5901 |
c-Di-AMP sodium
salt |
A2A inverse
agonist; also endogenous STING and DDX41 agonist |
1063 |
CGS 21680
hydrochloride |
A2A agonist |
1710 |
CV 1808 |
Non-selective
adenosine A2 receptor agonist |
5147 |
Istradefylline |
Potent and
selective A2A antagonist |
4603 |
LUF 5834 |
Potent adenosine
A2A and A2B receptor partial agonist |
4334 |
PSB 0777 ammonium
salt |
Potent adenosine
A2A agonist |
2463 |
SCH 442416 |
Very selective,
high affinity A2A antagonist |
2270 |
SCH 58261 |
Potent, highly
selective A2A antagonist |
4407 |
TC-G 1004 |
Potent and
selective A2A antagonist |
1036 |
ZM 241385 |
Potent and highly
selective A2A antagonist |
|
|
|
Adenosine
A2B Receptor Agonists, Antagonist |
|
Cat. No. |
Product |
Activity |
4472 |
BAY 60-6583 |
Potent partial A2B
agonist; cardioprotective |
7954 |
CELT-327 |
Potent and
selective hA2B/A3 adenosine receptor fluorescent antagonist |
1710 |
CV 1808 |
Non-selective
adenosine A2 receptor agonist |
4727 |
GS 6201 |
Selective A2B
antagonist |
6787 |
KI-7 |
Positive allosteric
modulator of A2B receptors |
4603 |
LUF 5834 |
Potent adenosine
A2A and A2B receptor partial agonist |
2752 |
MRS 1754 |
Selective A2B
antagonist |
3199 |
PSB 0788 |
Selective A2B
antagonist |
2009 |
PSB 1115 |
Selective human A2B
antagonist; water-soluble |
3198 |
PSB 603 |
Highly selective
A2B antagonist |
|
|
|
Adenosine
A3 Receptor Agonists, Antagonist |
|
Cat. No. |
Product |
Activity |
1104 |
2-Cl-IB-MECA |
Highly selective A3
agonist |
7954 |
CELT-327 |
Potent and
selective hA2B/A3 adenosine receptor fluorescent antagonist |
7628 |
DPTN |
Potent and
selective A3 adenosine receptor antagonist |
1579 |
HEMADO |
High affinity
selective A3 agonist |
1066 |
IB-MECA |
A3 selective
agonist |
1217 |
MRS 1220 |
Highly potent and
selective hA3 antagonist |
1385 |
MRS 1334 |
Potent, highly
selective hA3 antagonist |
5428 |
MRS 5698 |
High affinity and
selective A3 agonist |
2010 |
PSB 10
hydrochloride |
Potent, highly
selective hA3 receptor antagonist/inverse agonist |