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 ǰȳ  Ű   Pharmacology

Retinoid Receptor Small Molecules

Retinoid Receptor ʿ Small Molecules Ұմϴ.

TOCRIS
ǰ ϱ
μϱ





Agonists
Cat. No. Product Name / Activity
4046 AC 261066
RARβ2 agonist
2436 AC 55649
Selective RARβ2 agonist
2852 Adapalene
RARβ and RARγ agonist
760 AM 580
Retinoic acid analog; RARα agonist
3507 AM 80
RARα agonist; anticancer agent
3505 BMS 753
RARα-selective agonist
3410 BMS 961
Selective RARγ agonist
2554 CD 1530
Potent and selective RARγ agonist
3824 CD 2314
Selective RARβ agonist
1549 CD 437
RARγ-selective agonist
2020 Ch 55
Potent RAR agonist
695 Retinoic acid
Endogenous retinoic acid receptor agonist
3997 Tazarotene
Receptor-selective retinoid; binds RAR-β and -γ
761 TTNPB
Retinoic acid analog; RAR agonist
Inverse Agonists
Cat. No. Product Name / Activity
3509 BMS 493
Pan-RAR inverse agonist
Antagonists
Cat. No. Product Name / Activity
5758 AGN 193109
High affinity pan-RAR antagonist
3660 BMS 195614
Selective RARα antagonist
3800 CD 2665
Selective RARβ/γ antagonist
3823 ER 50891
Selective RARα antagonist
2021 LE 135
Selective RARβ antagonist
5984 LY 2955303
High affinity and selective RARγ antagonist
3822 MM 11253
RARγ-selective antagonist
Others
Cat. No. Product Name / Activity
3409 BMS 453
Synthetic retinoid and RARβ agonist; also RARα and RARγ antagonist
5849 EC 19
Synthetic retinoid; induces differentiation of stem cells
4011 EC 23
Synthetic retinoid; induces differentiation of stem cells
1396 Fenretinide
Synthetic retinoid; antiproliferative and antioxidant
2705 Liarozole dihydrochloride
Blocks retinoic acid metabolism



Agonists
Cat. No. Product Name / Activity
5868 SR 0987
T cell-specific RORγ (RORγt) agonist
4874 SR 1078
RORα/γ agonist
Inverse Agonists
Cat. No. Product Name / Activity
5987 (±)-ML 209
RORγt inverse agonist; suppresses Th17 cell differentiation
4868 SR 1001
RORα/γ inverse agonist
4869 SR 2211
Selective RORγ inverse agonist
Antagonists
Cat. No. Product Name / Activity
6223 XY 018
RORγ antagonist; inhibits AR expression
Others
Cat. No. Product Name / Activity
0695 Retinoic acid
Endogenous retinoic acid receptor agonist; proposed RORβ ligand



Agonists
Cat. No. Product Name / Activity
5819 Bexarotene
Potent and selective RXR agonist
3302 CD 3254
Potent and selective RXRα agonist
3687 Docosahexaenoic acid
RXR agonist
4064 Fluorobexarotene
RXR agonist
5920 LG 100268
Potent and selective RXR agonist; also activates RXR/PPARγ heterodimers
0695 Retinoic acid
Endogenous retinoic acid receptor agonist
3411 SR 11237
Pan RXR agonist
Antagonists
Cat. No. Product Name / Activity
3912 HX 531
Potent RXR antagonist
5086 PA 452
RXR antagonist
3303 UVI 3003
RXR antagonist
Modulators
Cat. No. Product Name / Activity
3508 LG 101506
Selective RXR modulator
Others
Cat. No. Product Name / Activity
1396 Fenretinide
Synthetic retinoid; antiproliferative and antioxidant
3913 HX 630
RXR synergist
3831 LG 100754
RXR:PPAR agonist
2705 Liarozole dihydrochloride
Blocks retinoic acid metabolism