Peptide Hormone Receptor Small Molecules


Peptide Hormone Receptor 연구에 필요한 Small Molecules을 소개합니다.
		TOCRIS

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	Agonists
	Cat. No.	Product Name / Activity
	5600	BA 1
		Potent bombesin agonist
	2716	BIM 187
		Bombesin/GRP receptor agonist
	1149	Bombesin
		Involved in gastrointestinal tract function
	1789	GRP (human)
		Endogenous GRP receptor agonist
	1788	GRP (porcine)
		Endogenous GRP receptor agonist

	Antagonists
	Cat. No.	Product Name / Activity
	2717	BIM 189
		Bombesin antagonist
	3237	BIM 23042
		Selective neuromedin B receptor antagonist (NMB-R, BB1)
	3422	[D-Phe12,Leu14]-Bombesin
		Bombesin receptor antagonist
	5599	ML 18
		BRS-3 antagonist; also GRPR agonist
	2602	PD 176252
		GRP (BB2) and NMB (BB1) receptor antagonist

	Others
	Cat. No.	Product Name / Activity
	1893	Alytesin
		Amphibian bombesin-like peptide
	1916	Litorin
		Amphibian bombesin-like peptide
	1908	Neuromedin B (porcine)
		Mammalian bombesin-like peptide

	Agonists
	Cat. No.	Product Name / Activity
	2257	GIP (1-39)
		Highly potent insulinotropic peptide; GIP agonist
	2084	GIP (human)
		Potent insulinotropic gut hormone; GIP agonist
	6699	[D-Ala2]-GIP (human)
		Highly potent GIP agonist
	5837	[Pro3]-GIP (Rat)
		High affinity rat GIP partial agonist

	Antagonists
	Cat. No.	Product Name / Activity
	5838	[Pro3]-GIP (Mouse)
		GIP receptor antagonist

	Agonists
	Cat. No.	Product Name / Activity
	1463	Ghrelin (human)
		Endogenous ghrelin receptor agonist
	1465	Ghrelin (rat)
		Endogenous ghrelin receptor agonist
	2261	L-692,585
		Potent, non-peptide ghrelin receptor agonist
	5272	MK 0677
		High affinity ghrelin receptor agonist
	2308	Tabimorelin hemifumarate
		Potent, orally active ghrelin receptor agonist

	Inverse Agonists
	Cat. No.	Product Name / Activity
	5830	K-(D-1-Nal)-FwLL-NH2
		High affinity and potent ghrelin receptor inverse agonist
	6347	PF 04628935
		Potent ghrelin receptor inverse agonist
	6350	PF 05190457
		High affinity and selective ghrelin receptor inverse agonist
	1946	[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
		Potent ghrelin receptor inverse agonist; Antagonist at other neuropeptide receptors

	Antagonists
	Cat. No.	Product Name / Activity
	1922	[D-Lys3]-GHRP-6
		Ghrelin receptor antagonist
	3959	YIL 781
		Ghrelin receptor (GHS-R1a) antagonist

	Others
	Cat. No.	Product Name / Activity
	3374	Cortistatin 14
		Endogenous neuropeptide; binds ghrelin receptor and sst1 - sst5
	2951	[Des-octanoyl]-Ghrelin (rat)
		Major circulating form of ghrelin; devoid of activity at GHS receptor
	1346	des-Gln14-Ghrelin (rat)
		Endogenous ghrelin receptor ligand
	2260	[Des-octanoyl]-Ghrelin (human)
		Major circulating form of ghrelin; devoid of activity at ghrelin receptor but is active in vivo
	5560	Obestatin (human)
		Endogenous anorexigenic peptide; opposes actions of ghrelin
	2445	Obestatin (rat)
		Endogenous anorexigenic peptide; opposes actions of ghrelin

	Agonists
	Cat. No.	Product Name / Activity
	1933	Exendin-4
		Potent GLP-1 receptor agonist
	5374	GLP-1 (7-37)
		Endogenous bioactive GLP-1 receptor ligand
	1851	Glucagon-like peptide 1 (1-37) (human, rat)
		Endogenous pancreatic peptide
	2082	Glucagon-like peptide 1 (7-36) amide (human, rat)
		Potent insulinotropic peptide
	6517	Liraglutide
		Highly potent, long-acting GLP-1 receptor agonist
	2094	Oxyntomodulin (porcine, bovine)
		GLP-1 receptor agonist; endogenous preproglucagon derived peptide; modulates feeding and metabolism

	Antagonists
	Cat. No.	Product Name / Activity
	2081	Exendin-3 (9-39) amide
		Potent GLP-1 receptor antagonist
	3266	GLP-1 (9-36) amide
		Metabolite of GLP-1-(7-36) (Cat. No. 2082)
	6355	VU 0650991
		Non-competitive GLP-1 antagonist; orally bioavailable and brain penetrant

	Modulators
	Cat. No.	Product Name / Activity
	4778	BETP
		Positive allosteric modulator of GLP-1 receptors

	Agonists
	Cat. No.	Product Name / Activity
	6927	Glucagon (Human, Porcine)
		Endogenous glucagon receptor agonist

	Antagonists
	Cat. No.	Product Name / Activity
	2216	des-His1-[Glu9]-Glucagon (1-29) amide
		Glucagon receptor antagonist
	2311	L-168,049
		Potent, orally active human glucagon receptor antagonist

	Others
	Cat. No.	Product Name / Activity
	2094	Oxyntomodulin (porcine, bovine)
		Endogenous gut peptide; modulates feeding and metabolism

	Agonists
	Cat. No.	Product Name / Activity
	1918	Secretin (human)
		Gastrointestinal peptide
	1919	Secretin (rat)
		Gastrointestinal peptide

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