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Pharmacology

Opioid Receptor Small Molecules


Opiod receptor에 대한 small molecule을 소개합니다.
		TOCRIS

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	Agonists
	Cat. No.	Product Name / Activity
	4335	AR-M 1000390 hydrochloride
		Low-internalizing δ agonist
	1663	BW 373U86
		Potent, selective non-peptide δ agonist
	3790	DADLE
		Prototypical δ agonist
	4591	Deltorphin I
		Potent δ agonist
	1180	[D-Ala2]-Deltorphin II
		Selective δ agonist peptide
	1431	DPDPE
		Selective δ agonist
	2962	6'-GNTI dihydrochloride
		Selective κ/δ opioid heterodimer receptor agonist
	0921	SB 205607 dihydrobromide
		Selective, high affinity non-peptide δ1 agonist
	1529	SNC 162
		Potent, selective non-peptide δ agonist
	0764	SNC 80
		Highly selective non-peptide δ agonist

	Antagonists
	Cat. No.	Product Name / Activity
	0754	N-Benzylnaltrindole hydrochloride
		Selective non-peptide δ2 antagonist
	0899	BNTX maleate
		Standard δ1 selective antagonist
	0827	ICI 154,129
		δ selective peptide antagonist
	0820	ICI 174,864
		δ selective peptide antagonist
	0892	Naltriben mesylate
		Standard δ2 selective antagonist
	1410	SDM25N hydrochloride
		Potent, selective non-peptide δ antagonist; also inhibits dengue virus replication
	6729	TAN 452
		Potent and selective peripherally acting δ opioid antagonist; antianalgesic.

	Modulators
	Cat. No.	Product Name / Activity
	5983	BMS 986187
		Potent positive allosteric modulator of δ receptors

	Agonists
	Cat. No.	Product Name / Activity
	0699	BRL 52537 hydrochloride
		Potent and selective κ agonist
	3195	Dynorphin A
		Endogenous κ agonist
	3196	Dynorphin B
		Endogenous κ agonist
	2962	6'-GNTI dihydrochloride
		Selective κ/δ opioid heterodimer receptor agonist
	1483	GR 89696 fumarate
		Subtype-selective κ agonist
	0778	ICI 199,441 hydrochloride
		Potent κ agonist
	0822	ICI 204,448 hydrochloride
		κ agonist, acts peripherally
	0783	N-MPPP Hydrochloride
		Selective κ agonist
	5519	(-)-Pentazocine
		κ-agonist; antinociceptive
	2134	Salvinorin A
		Highly potent and selective κ agonist
	0471	(+)-U-50488 hydrochloride
		Selective κ agonist; less active enantiomer of (±)-U-50488 (Cat. No. 0495)
	0495	(±)-U-50488 hydrochloride
		Selective κ agonist
	0496	(-)-U-50488 hydrochloride
		Selective κ agonist; more active enantiomer of (±)-U-50488 (Cat. No. 0495)

	Antagonists
	Cat. No.	Product Name / Activity
	0347	nor-Binaltorphimine dihydrochloride
		Selective κ antagonist
	0794	DIPPA hydrochloride
		Selective and irreversible κ antagonist
	1282	GNTI dihydrochloride
		Potent, selective κ antagonist
	4866	ML 190
		Selective κ opioid receptor antagonist

	Others
	Cat. No.	Product Name / Activity
	5611	Salvinorin B
		Activates the κ-opioid DREADD (KORD)

	Agonists
	Cat. No.	Product Name / Activity
	1171	DAMGO
		Selective μ agonist
	1055	Endomorphin-1
		Potent and selective μ agonist
	1056	Endomorphin-2
		Potent and selective μ agonist
	0840	Loperamide hydrochloride
		Peripherally acting μ agonist; Ca2+ channel blocker
	3636	Meptazinol hydrochloride
		μ1 partial agonist
	2024	PL 017
		Selective μ agonist
	3848	Sinomenine hydrochloride
		μ agonist; antinociceptive and anti-inflammatory

	Antagonists
	Cat. No.	Product Name / Activity
	0898	Clocinnamox mesylate
		Irreversible μ antagonist
	1560	CTAP
		Potent and selective μ antagonist
	1578	CTOP
		Potent and selective μ antagonist
	2601	Cyprodime hydrochloride
		Selective μ antagonist
	0926	β-Funaltrexamine hydrochloride
		Irreversible and selective μ antagonist
	6109	Methylnaltrexone bromide
		μ antagonist; peripherally restricted
	0591	Naloxonazine dihydrochloride
		Selective μ1 antagonist

	Agonists
	Cat. No.	Product Name / Activity
	2808	Buprenorphine hydrochloride
		NOP agonist; also displays mixed action δ, κ and μ receptors
	3763	MCOPPB trihydrochloride
		Potent NOP receptor agonist
	1780	NNC 63-0532
		Potent non-peptide NOP agonist; brain penetrant
	0910	Nociceptin
		Endogenous NOP agonist
	1590	[Arg14,Lys15]Nociceptin
		Highly potent and selective NOP agonist
	1566	[(pF)Phe4]Nociceptin(1-13)NH2
		Potent, selective nociceptin receptor agonist
	1092	[Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2
		Selective nociceptin receptor agonist
	3932	Orphanin FQ (1-11)
		Potent NOP agonist; displays analgesic properties
	1387	Ac-RYYRWK-NH2
		Potent, selective NOP partial agonist peptide
	3240	SCH 221510
		Potent and selective NOP agonist

	Antagonists
	Cat. No.	Product Name / Activity
	3661	BAN ORL 24
		Potent and selective NOP antagonist
	2598	(±)-J 113397
		Potent and selective NOP antagonist
	2481	JTC 801
		Selective NOP antagonist
	1308	[Nphe1]Nociceptin(1-13)NH2
		Selective, competitive nociceptin antagonist
	1118	Nocistatin (bovine)
		Opposes action of nociceptin
	1198	Nocistatin (human)
		Human putative counterpart of nocistatin
	3573	SB 612111 hydrochloride
		Selective NOP antagonist
	2508	Trap 101
		Potent and selective NOP antagonist; active in vivo
	1552	UFP-101
		Potent, selective silent antagonist for NOP

	Ligand
	Cat. No.	Product Name / Activity
	1239	Ac-RYYRIK-NH2
		High affinity NOP ligand

	Others
	Cat. No.	Product Name / Activity
	1266	Nociceptin (1-7)
		Bioactive metabolite of nociceptin
	1119	NocII
		Orphan neuropeptide