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 ǰȳ  Ű   Pharmacology

Cannabinoid Receptor Small Molecules

Cannabinoid Receptor agonist & antagonist Ұմϴ.

TOCRIS
ǰ ϱ
μϱ




Agonists
Cat. No. Product Name / Activity
1319 ACEA
Potent and highly selective CB1 agonist
1318 ACPA
Potent and selective CB1 agonist
1781 ACPA (in Tocrisolve™ 100)
Potent and selective CB1 agonist; supplied in water-soluble emulsion
1354 Arvanil
Potent CB1 agonist; also anandamide transport inhibitor and TRPV1 agonist
1485 DEA
Endogenous CB1 agonist
2139 Leelamine hydrochloride
CB1 agonist
1121 (R)-(+)-Methanandamide
Potent and selective CB1 agonist
1782 (R)-(+)-Methanandamide (in Tocrisolve™ 100)
Potent and selective CB1 agonist; supplied in water-soluble emulsion
1568 NADA
Endogenous CB1 agonist; also vanilloid agonist and inhibitor of FAAH and AMT
1411 Noladin ether
Endogenous agonist for CB1 and GPR55
0878 Oleamide
CB1 agonist
3744 RVD-Hpα
Selective CB1 agonist; also CB2 PAM
Inverse Agonists
Cat. No. Product Name / Activity
1115 AM 281
Potent and selective CB1 inverse agonist
3791 Hemopressin (human, mouse)
Selective CB1 inverse agonist
1764 Hemopressin (rat)
Selective CB1 inverse agonist
2387 LY 320135
Selective CB1 inverse agonist
0923 SR 141716A
Selective CB1 inverse agonist
4345 TC-C 14G
High affinity and potent CB1 inverse agonist
Antagonists
Cat. No. Product Name / Activity
1117 AM 251
Potent CB1 antagonist; also GPR55 agonist
6193 AM 4113
High affinity and selective CB1 antagonist
5443 AM 6545
High affinity and selective CB1 antagonist
6763 AVE 1625
Potent and selective CB1 receptor antagonist
4236 CP 945598 hydrochloride
CB1 antagonist
4063 MJ 15
Potent and selective CB1 antagonist
5746 NESS 0327
Ultra-high affinity and selective CB1 antagonist
3676 PF 514273
High affinity and selective CB1 antagonist
4605 (±)-SLV 319
High affinity and selective CB1 antagonist
Modulators
Cat. No. Product Name / Activity
2957 Org 27569
Potent allosteric modulator of CB1 receptors
5321 PSNCBAM-1
Negative allosteric modulator of CB1 receptors
Others
Cat. No. Product Name / Activity
1655 O-2050
Putative CB1 antagonist; displays mixed activity at CB receptors
2540 Tocrifluor T1117
Fluorescent cannabinoid ligand; fluorescent form of AM 251 (Cat. No. 1117)



Agonists
Cat. No. Product Name / Activity
2663 CB 65
High affinity, selective CB2 agonist
2678 GP 2a
Selective CB2 agonist
2374 GW 405833
Selective, high affinity CB2 receptor partial agonist
3088 HU 308
Potent and selective CB2 agonist
1341 JWH 015
Selective CB2 agonist
1343 JWH 133
Potent and selective CB2 agonist
5826 LEI 101 hydrochloride
Potent and selective CB2 partial agonist; orally biovailable
4205 MDA 19
CB2 agonist
6220 PM 226
Potent and selective CB2 receptor agonist; BBB permeable; neuroprotective
3556 SER 601
Potent, selective CB2 agonist
Inverse Agonists
Cat. No. Product Name / Activity
1120 AM 630
Selective CB2 inverse agonist
4756 COR 170
Selective CB2 receptor inverse agonist
2764 GP 1a
CB2 receptor inverse agonist
2479 JTE 907
Selective CB2 receptor inverse agonist
5815 SCH 336
Highly potent and selective CB2 inverse agonist
5039 SR 144528
High affinity and selective CB2 inverse agonist
Modulators
Cat. No. Product Name / Activity
6832 Ec2la
Positive allosteric modulator of CB2 receptors; active in vivo
3744 RVD-Hpα
High affinity CB2 positive allosteric modulator; also CB1 agonist