• Home
  • About us
  • Log-In
  • Join Us
  • Sitemap
  • Recruit
ǰ/ Q&A
ֹ
Խ
ڷû
ڷ
Ŭ
A/S
Ŭ ȸ
 ǰȳ  Ű   Pharmacology

Adenosine Receptors Small molecules

Adenosine Receptor ʿ Small molecules Ұմϴ.

TOCRIS
ǰ ϱ
μϱ





Agonists
Cat. No. Product Name / Activity
1705 2-Chloro-N6-cyclopentyladenosine
Potent, selective A1 agonist
1702 N6-Cyclopentyladenosine
Potent, selective A1 agonist
5122 Dansyl-NECA
Potent and selective fluorescent adenosine A1 agonist
3576 (±)-5'-Chloro-5'-deoxy-ENBA
Highly selective A1 agonist
1957 GR 79236
A1 agonist
2281 2'-MeCCPA
Very selective and potent A1 receptor agonist
2465 SDZ WAG 994
Potent, selective A1 agonist
Inverse Agonists
Cat. No. Product Name / Activity
5351 PQ 69
Potent and selective A1 inverse agonist
Antagonists
Cat. No. Product Name / Activity
6137 8-Cyclopentyl-1,3-dimethylxanthine
High affinity adenosine A1 receptor antagonist
0486 1,3-Dipropyl-8-phenylxanthine
A1 selective antagonist
0439 DPCPX
A1 selective antagonist
4167 KW 3902
Selective A1 antagonist
2019 PSB 36
Potent and selective A1 antagonist
3344 SLV 320
Potent and selective A1 antagonist
Modulators
Cat. No. Product Name / Activity
1363 PD 81723
Allosteric potentiator of A1 receptors



Agonists
Cat. No. Product Name / Activity
1063 CGS 21680 hydrochloride
A2A agonist
1710 CV 1808
Non-selective adenosine A2 receptor agonist
4603 LUF 5834
Potent adenosine A2A and A2B receptor partial agonist
4334 PSB 0777 ammonium salt
Potent adenosine A2A agonist
Inverse Agonists
Cat. No. Product Name / Activity
5901 c-Di-AMP sodium salt
A2A inverse agonist; also endogenous STING and DDX41 agonist
Antagonists
Cat. No. Product Name / Activity
3937 ANR 94
Adenosine A2A antagonist
3306 8-(3-Chlorostyryl)caffeine
Selective A2A antagonist. Also MAO-B inhibitor
5147 Istradefylline
Potent and selective adenosine A2A receptor antagonist
4783 Lu AA 47070
Prodrug of a potent and selective adenosine A2A receptor antagonist
2463 SCH 442416
Very selective, high affinity A2A antagonist
2270 SCH 58261
Potent, highly selective A2A antagonist
4407 TC-G 1004
Potent and selective A2A antagonist
1036 ZM 241385
Potent, highly selective A2A antagonist


Agonists
Cat. No. Product Name / Activity
4472 BAY 60-6583
Potent A2B receptor agonist; cardioprotective
1710 CV 1808
Non-selective adenosine A2 receptor agonist
4603 LUF 5834
Potent adenosine A2A and A2B receptor partial agonist
Inverse Agonists
Cat. No. Product Name / Activity
1584 MRS 1706
Potent and selective A2B inverse agonist
Agonists
Cat. No. Product Name / Activity
4727 GS 6201
Selective A2B antagonist
5965 ISAM 140
High affinity A2B receptor antagonist
2752 MRS 1754
Selective A2B antagonist
3199 PSB 0788
Selective A2B antagonist
2009 PSB 1115
Selective human A2B receptor antagonist; water-soluble
3198 PSB 603
Highly selective A2B antagonist
Modulators
Cat. No. Product Name / Activity
6787 KI-7
Positive allosteric modulator of A2B receptors


Agonists
Cat. No. Product Name / Activity
1104 2-Cl-IB-MECA
Highly selective A3 agonist
1579 HEMADO
High affinity selective A3 agonist
1066 IB-MECA
A3 selective agonist
5428 MRS 5698
High affinity and selective A3 adenosine receptor agonist
Antagonists
Cat. No. Product Name / Activity
4041 MRE 3008F20
Highly potent and selective adenosine A3 receptor antagonist
1217 MRS 1220
Highly potent, selective hA3 antagonist
1385 MRS 1334
Potent, highly selective hA3 antagonist
2010 PSB 10 hydrochloride
Potent, highly selective hA3 receptor antagonist/inverse agonist
2012 PSB 11 hydrochloride
Potent, selective hA3 receptor antagonist/inverse agonist
1359 VUF 5574
Potent, selective hA3 antagonist